Somatropin

Generic Details

Generic Name

Somatropin

Other Names

  • Human Growth Hormone
  • HGH

Drug Class

  • Hormone
  • Growth Promoter

Chemical Formula

C990H1529N263O299S7

Molecular Weight

22,125.0 g/mol

Mechanism of Action

  • Stimulates growth and cell reproduction

Indications

  • Pediatric growth hormone deficiency
  • Turner syndrome
  • Chronic kidney disease
  • Muscle wasting in HIV/AIDS
  • Short bowel syndrome

Common Dosage Forms

  • Injection

Typical Dosage

  • 0.1-0.3 mg/kg/day

Pediatric Dosage

  • Varies based on weight and condition, typically starting at 0.1 mg/kg/day

Geriatric Dosage

  • Dose adjustment may be necessary based on individual response

Side Effects

  • Headache
  • Nausea
  • Joint pain
  • Edema
  • Hypertension
  • Hyperglycemia

Contraindications

  • Active malignancy
  • Acute critical illness

Pregnancy Category

  • Category B

Lactation Safety

  • Compatible with breastfeeding, monitor for growth in infant

Drug Interactions

  • Insulin
  • Oral hypoglycemic agents
  • Corticosteroids

Overdose Symptoms

  • Hypoglycemia
  • Edema
  • Carpal tunnel syndrome

Antidote for Overdose

  • Symptomatic and supportive treatment

Storage Conditions

  • Refrigerate at 2-8°C, do not freeze

Pharmacokinetics

  • Absorption: Rapid and complete after subcutaneous injection
  • Distribution: Mainly in the liver, kidney, and muscle tissues
  • Metabolism: Metabolized in the liver
  • Excretion: Primarily excreted in the urine

Precautions

  • Monitor glucose levels in diabetic patients
  • Monitor thyroid function in patients with hypothyroidism

Warnings

  • Increased risk of intracranial hypertension in pediatric patients with Prader-Willi syndrome
  • Monitor for signs of leukemia in patients with short stature due to chronic renal insufficiency

Others

  • Somatropin should not be used for growth promotion in children with closed epiphyses