Bambuterol Hydrochloride

Generic Details

Generic Name

Bambuterol Hydrochloride

Other Names

  • Bambuterol HCl

Drug Class

  • Bronchodilator
  • Beta-2 Agonist

Chemical Formula

C18H29N3O4

Molecular Weight

347.44 g/mol

Mechanism of Action

  • Selective β2-adrenergic agonist
  • Prodrug of terbutaline

Indications

  • Chronic obstructive pulmonary disease (COPD)
  • Asthma

Common Dosage Forms

  • Tablet
  • Syrup

Typical Dosage

  • 10-20 mg once daily

Pediatric Dosage

  • Consult pediatrician for appropriate dosage

Geriatric Dosage

  • Adjust dosage based on renal function

Side Effects

  • Tremors
  • Tachycardia
  • Hypokalemia
  • Headache

Contraindications

  • Hypersensitivity to beta-adrenergic agonists

Pregnancy Category

  • C - Risk cannot be ruled out

Lactation Safety

  • Limited data, use caution

Drug Interactions

  • Beta-blockers
  • Diuretics

Overdose Symptoms

  • Severe tremors
  • Palpitations
  • Hypotension

Antidote for Overdose

  • Beta-blockers

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Well absorbed orally
  • Distribution: Wide distribution in the body
  • Metabolism: Metabolized in the liver
  • Excretion: Primarily excreted in urine

Precautions

  • Monitor potassium levels
  • Caution in patients with cardiovascular disease

Warnings

  • Not to be used as a rescue medication for acute bronchospasm

Others