Tetracycline Hydrochloride (Oral)

Generic Details

Generic Name

Tetracycline Hydrochloride Oral

Other Names

  • Tetracycline HCl

Drug Class

  • Antibiotic
  • Tetracycline

Chemical Formula

C22H24N2O8.HCl

Molecular Weight

480.9 g/mol

Mechanism of Action

  • Inhibits bacterial protein synthesis by binding to the 30S ribosomal subunit

Indications

  • Acne
  • Chlamydia infection
  • Mycoplasma pneumonia
  • Lyme disease
  • Gonorrhea

Common Dosage Forms

  • Capsule
  • Tablet

Typical Dosage

  • 250 mg every 6 hours

Pediatric Dosage

  • 2-4 mg/kg/dose every 6 hours

Geriatric Dosage

  • Lower doses may be required due to decreased renal function

Side Effects

  • Nausea
  • Vomiting
  • Diarrhea
  • Photosensitivity
  • Tooth discoloration
  • Esophageal irritation

Contraindications

  • Pregnancy
  • Children under 8 years old
  • Severe liver disease

Pregnancy Category

  • D

Lactation Safety

  • Not recommended, can pass into breast milk and harm the infant

Drug Interactions

  • Antacids containing aluminum, calcium, or magnesium reduce tetracycline absorption
  • Penicillins may reduce effectiveness of tetracycline

Overdose Symptoms

  • Nausea
  • Vomiting
  • Diarrhea
  • Increased intracranial pressure

Antidote for Overdose

No specific antidote, treatment is symptomatic

Storage Conditions

  • Store at room temperature away from light and moisture

Pharmacokinetics

  • Absorption: Well absorbed orally
  • Distribution: Distributed widely in body tissues
  • Metabolism: Metabolized in the liver
  • Excretion: Excreted in urine and feces

Precautions

  • Avoid sunlight and UV light exposure due to photosensitivity
  • Take on an empty stomach to enhance absorption
  • Do not take with dairy products, antacids, or iron supplements

Warnings

  • May cause permanent tooth discoloration in children under 8 years old
  • Can lead to overgrowth of non-susceptible organisms such as fungi

Others

  • Tetracycline should not be taken with food, as it can reduce absorption.