Beclomethasone Dipropionate (Inhaler)
Generic Details
Generic Name
Beclomethasone Dipropionate Inhaler
Other Names
- Qvar
- Becotide
- Vanceril
Drug Class
- Corticosteroid
Chemical Formula
C28H37ClO7
Molecular Weight
521.04 g/mol
Mechanism of Action
- Anti-inflammatory effects by inhibiting the release of inflammatory mediators.
Indications
- Asthma
- Chronic obstructive pulmonary disease (COPD)
Common Dosage Forms
- Inhaler
Typical Dosage
- 100-200 mcg twice daily for asthma maintenance therapy
Pediatric Dosage
- Children: 50-100 mcg twice daily
Geriatric Dosage
- Use with caution, dosing may need adjustment based on individual factors.
Side Effects
- Throat irritation
- Hoarseness
- Fungal infections in the mouth/throat
- Increased risk of pneumonia
Contraindications
- Hypersensitivity to beclomethasone or any components of the formulation
Pregnancy Category
- C - Use with caution if benefits outweigh risks
Lactation Safety
- Caution advised as it can pass into breast milk
Drug Interactions
- Caution with strong CYP3A4 inhibitors (e.g., ritonavir) may increase systemic corticosteroid effects.
Overdose Symptoms
- Nausea
- Vomiting
- Headache
- Dizziness
Antidote for Overdose
- Supportive care and monitoring
Storage Conditions
- Store at controlled room temperature between 68°F to 77°F (20°C to 25°C). Protect from light.
Pharmacokinetics
- Absorption: Rapidly absorbed from the lungs
- Distribution: Mainly to the lungs
- Metabolism: Hepatic metabolism
- Excretion: Primarily eliminated in the feces
Precautions
- Monitor for signs of adrenal insufficiency with long-term use
- Gradually taper doses when discontinuing therapy to prevent adrenal crisis
Warnings
- Not for acute asthma attacks, requires regular daily use for optimal effect
Others
- Always rinse mouth after inhalation to reduce the risk of oral fungal infections.