Levothyroxine Sodium

Generic Details

Generic Name

Levothyroxine-sodium

Other Names

  • Synthroid
  • Levoxyl
  • Eltroxin

Drug Class

  • Thyroid hormone

Chemical Formula

C15H10I4NNaO4

Molecular Weight

798.85 g/mol

Mechanism of Action

  • Acts as a synthetic form of thyroxine (T4) which is converted to triiodothyronine (T3) in the body. It regulates metabolic processes and influences the growth and development of tissues.

Indications

  • Hypothyroidism
  • Thyroid cancer (after thyroidectomy)

Common Dosage Forms

  • Tablet
  • Capsule

Typical Dosage

  • 25-200 mcg once daily in the morning on an empty stomach

Pediatric Dosage

  • Dose varies based on weight and age, consult a healthcare provider

Geriatric Dosage

  • Lower starting doses may be required for the elderly

Side Effects

  • Palpitations
  • Weight loss
  • Tremors
  • Headache
  • Nervousness

Contraindications

  • Untreated thyrotoxicosis
  • Acute myocardial infarction
  • Uncorrected adrenal insufficiency

Pregnancy Category

  • A

Lactation Safety

  • Considered safe while breastfeeding

Drug Interactions

  • Warfarin
  • Phenytoin
  • Digoxin

Overdose Symptoms

  • Chest pain
  • Increased heart rate
  • Fever
  • Excessive sweating

Antidote for Overdose

  • Activated charcoal
  • Cholestyramine

Storage Conditions

  • Store at room temperature below 25°C (77°F)

Pharmacokinetics

  • Absorption: Absorbed in the upper small intestine
  • Distribution: Mainly bound to serum proteins
  • Metabolism: Liver
  • Excretion: Primarily in urine

Precautions

  • Dose adjustments may be needed in patients with cardiovascular disease or diabetes

Warnings

  • Regular monitoring of thyroid function tests is essential during treatment

Others