Diclofenac Potassium

Generic Details

Generic Name

Diclofenac-Potassium

Other Names

  • Diclofenac K
  • Potassium Diclofenac

Drug Class

  • Nonsteroidal anti-inflammatory drug (NSAID)

Chemical Formula

C14H10Cl2KNO2

Molecular Weight

334.24 g/mol

Mechanism of Action

  • Inhibits prostaglandin synthesis by blocking cyclooxygenase enzymes (COX-1 and COX-2)

Indications

  • Pain relief
  • Inflammation reduction
  • Fever reduction

Common Dosage Forms

  • Tablet
  • Capsule
  • Topical gel
  • Eye drops

Typical Dosage

  • 50 mg to 150 mg per day in divided doses

Pediatric Dosage

  • Consult pediatrician for appropriate dosage

Geriatric Dosage

  • Lower starting dose may be required for elderly patients

Side Effects

  • Stomach ulcers
  • Gastrointestinal bleeding
  • Kidney problems
  • Liver toxicity
  • Headache
  • Dizziness
  • Rash

Contraindications

  • History of allergic reaction to NSAIDs
  • Active peptic ulcer disease
  • Severe heart failure

Pregnancy Category

  • Category C: Consult healthcare provider before use

Lactation Safety

  • Limited data available - use caution and consult healthcare provider

Drug Interactions

  • Aspirin
  • Warfarin
  • ACE Inhibitors
  • Diuretics

Overdose Symptoms

  • Nausea
  • Vomiting
  • Stomach pain
  • Drowsiness
  • Seizures

Antidote for Overdose

  • Activated charcoal
  • Supportive care

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Well absorbed from the gastrointestinal tract
  • Distribution: Highly protein-bound
  • Metabolism: Undergoes hepatic metabolism
  • Excretion: Primarily excreted in the urine

Precautions

  • Use with caution in patients with a history of asthma
  • Monitor for signs of gastrointestinal bleeding or ulceration

Warnings

  • Increased risk of cardiovascular events
  • May cause serious gastrointestinal adverse events

Others

  • Avoid prolonged exposure to sunlight while using topical diclofenac preparations