Salbutamol

Generic Details

Generic Name

Salbutamol

Other Names

  • Albuterol

Drug Class

  • Beta2-adrenergic agonist

Chemical Formula

C13H21NO3

Molecular Weight

239.31 g/mol

Mechanism of Action

  • Selective agonist at beta2-adrenergic receptors resulting in bronchodilation

Indications

  • Asthma
  • Chronic obstructive pulmonary disease (COPD)
  • Exercise-induced bronchospasm

Common Dosage Forms

  • Inhaler
  • Nebulizer solution
  • Tablet
  • Syrup

Typical Dosage

  • Inhaler: 90mcg per actuation, 2 puffs every 4-6 hours as needed

Pediatric Dosage

  • Dosing based on weight and age, consult healthcare provider

Geriatric Dosage

  • Dosage adjustment may be needed, consult healthcare provider

Side Effects

  • Tachycardia
  • Tremor
  • Headache
  • Nervousness
  • Hypokalemia

Contraindications

  • Hypersensitivity to Salbutamol
  • Severe heart disease

Pregnancy Category

  • C

Lactation Safety

  • Compatible but monitor infant for side effects

Drug Interactions

  • Beta-blockers
  • Diuretics
  • Monoamine oxidase inhibitors

Overdose Symptoms

  • Palpitations
  • Tachycardia
  • Tremor
  • Hypokalemia

Antidote for Overdose

  • Beta-blockers

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Rapidly absorbed from the respiratory tract
  • Distribution: Widely distributed in the body
  • Metabolism: Primarily hepatic
  • Excretion: Mainly renal

Precautions

  • Use with caution in patients with cardiovascular disorders

Warnings

  • Do not exceed recommended dose
  • Seek medical help if symptoms worsen

Others

  • Available as a rescue inhaler for acute symptoms