Alpha Lipoic Acid

Generic Details

Generic Name

Alpha-Lipoic Acid

Other Names

  • Thioctic Acid
  • ALA

Drug Class

  • Antioxidant

Chemical Formula

C8H14O2S2

Molecular Weight

206.33 g/mol

Mechanism of Action

  • Acts as a cofactor for mitochondrial enzymes involved in energy metabolism
  • Regenerates antioxidants such as Vitamin C and Vitamin E

Indications

  • Diabetic neuropathy
  • Peripheral neuropathy
  • Antioxidant support

Common Dosage Forms

  • Oral tablets
  • Capsules

Typical Dosage

  • 600-1800mg per day in divided doses

Pediatric Dosage

  • Not established

Geriatric Dosage

  • Dosing adjustment may be needed based on renal function

Side Effects

  • Nausea
  • Vomiting
  • Rash
  • Hypoglycemia in diabetic patients

Contraindications

  • Hypersensitivity to Alpha-Lipoic Acid

Pregnancy Category

  • C

Lactation Safety

  • Not established, use with caution

Drug Interactions

  • Insulin and other antidiabetic medications
  • Thyroid medications

Overdose Symptoms

  • Hypoglycemia
  • Nausea
  • Vomiting

Antidote for Overdose

  • Supportive care and monitoring

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Well absorbed after oral administration
  • Distribution: Widely distributed in the body
  • Metabolism: Primarily metabolized in the liver
  • Excretion: Mainly excreted in the urine

Precautions

  • Monitor blood glucose levels in diabetic patients
  • Use with caution in patients with thyroid disorders

Warnings

  • Consult healthcare provider before use if pregnant or breastfeeding

Others

  • May improve insulin sensitivity in diabetic patients