Cefaclor Monohydrate

Generic Details

Generic Name

Cefaclor Monohydrate

Other Names

  • Cefaclor

Drug Class

  • Cephalosporin Antibiotic

Chemical Formula

C15H14ClN3O4S.H2O

Molecular Weight

385.82 g/mol

Mechanism of Action

  • Inhibits bacterial cell wall synthesis

Indications

  • Treatment of bacterial infections such as respiratory tract infections, urinary tract infections, skin and soft tissue infections, and otitis media

Common Dosage Forms

  • Capsules
  • Oral suspension

Typical Dosage

  • 250-500 mg every 8 hours for adults

Pediatric Dosage

  • 20 mg/kg/day in divided doses

Geriatric Dosage

  • Adjust dose based on renal function

Side Effects

  • Nausea
  • Vomiting
  • Diarrhea
  • Rash
  • Allergic reactions

Contraindications

  • Hypersensitivity to cephalosporins

Pregnancy Category

  • Category B - Safe for use during pregnancy

Lactation Safety

  • Compatible with breastfeeding

Drug Interactions

  • Probenecid - may increase cefaclor levels

Overdose Symptoms

  • Seizures
  • Encephalopathy

Antidote for Overdose

  • No specific antidote, treatment is symptomatic

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Well-absorbed orally
  • Distribution: Distributes well into tissues and fluids
  • Metabolism: Partially metabolized in the liver
  • Excretion: Excreted mainly through the kidneys

Precautions

  • Use with caution in patients with renal impairment

Warnings

  • May cause Clostridium difficile-associated diarrhea

Others

  • Complete the full course of treatment as prescribed