Cephalexin

Generic Details

Generic Name

Cephalexin

Other Names

  • Keflex
  • Ceporex

Drug Class

  • First-generation cephalosporin antibiotic

Chemical Formula

C16H17N3O4S

Molecular Weight

349.39 g/mol

Mechanism of Action

  • Inhibits bacterial cell wall synthesis by binding to penicillin-binding proteins

Indications

  • Treatment of skin and soft tissue infections
  • Respiratory tract infections
  • Urinary tract infections
  • Bone infections

Common Dosage Forms

  • Capsule
  • Tablet
  • Oral suspension

Typical Dosage

  • 250-500 mg every 6 hours

Pediatric Dosage

  • 25-50 mg/kg/day in divided doses

Geriatric Dosage

  • Dose adjustment may be required based on renal function

Side Effects

  • Nausea
  • Vomiting
  • Diarrhea
  • Rash
  • Hypersensitivity reactions

Contraindications

  • Hypersensitivity to cephalosporins
  • History of severe allergic reactions to penicillins

Pregnancy Category

  • Category B - Generally considered safe for use during pregnancy

Lactation Safety

  • Considered compatible with breastfeeding

Drug Interactions

  • Probenecid - may increase cephalexin levels

Overdose Symptoms

  • Nausea
  • Vomiting
  • Diarrhea

Antidote for Overdose

  • No specific antidote, supportive care

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Well absorbed orally
  • Distribution: Distributed widely in the body
  • Metabolism: Minimally metabolized
  • Excretion: Excreted unchanged in urine

Precautions

  • Use with caution in patients with renal impairment

Warnings

  • Potential for allergic reactions in patients with penicillin allergies

Others