Clobetasol Propionate
Generic Details
Generic Name
Clobetasol Propionate
Other Names
- Clobex
- Olux
- Temovate
Drug Class
- Corticosteroid
Chemical Formula
C25H32ClFO5
Molecular Weight
466.97 g/mol
Mechanism of Action
- It exerts its anti-inflammatory, antipruritic, and vasoconstrictive actions by binding to cytoplasmic glucocorticoid receptors.
Indications
- Psoriasis
- Eczema
- Dermatitis
- Lichen Planus
Common Dosage Forms
- Cream
- Ointment
- Solution
- Foam
Typical Dosage
- Apply a thin layer to the affected area once daily
Pediatric Dosage
- Consult healthcare provider for appropriate dosing
Geriatric Dosage
- May require lower doses due to increased risk of skin thinning and other side effects
Side Effects
- Skin irritation
- Burning
- Itching
- Dryness
- Redness
- Folliculitis
Contraindications
- Hypersensitivity to clobetasol propionate or any component of the formulation
Pregnancy Category
- Category C - Animal reproduction studies have shown an adverse effect on the fetus and there are no adequate and well-controlled studies in humans
Lactation Safety
- Use with caution, minimal amounts of corticosteroids may be absorbed and excreted in breast milk
Drug Interactions
- No significant drug interactions reported
Overdose Symptoms
- Topical corticosteroid overdose is rare but may lead to increased risk of systemic effects
Antidote for Overdose
- No specific antidote, treatment is symptomatic and supportive
Storage Conditions
- Store at controlled room temperature between 20°C to 25°C (68°F to 77°F)
Pharmacokinetics
- Absorption: Well absorbed through the skin
- Distribution: Protein binding is high
- Metabolism: Metabolized in the liver
- Excretion: Excreted mainly in the urine
Precautions
- Avoid use on the face, groin, or axillae unless directed by a healthcare provider
- Do not use occlusive dressings unless directed
Warnings
- Prolonged use may lead to skin atrophy
- Discontinue if no improvement is seen after a few weeks
Others
- Avoid abrupt discontinuation - taper off the medication slowly to prevent rebound effects