Norgestrel + Ethinyl Estradiol + Ferrous Fumarate

Generic Details

Generic Name

Norgestrel-Ethinyl-Estradiol-Ferrous Fumarate

Other Names

  • Combined Oral Contraceptive
  • Birth Control Pill

Drug Class

  • Combination Oral Contraceptive

Chemical Formula

C22H28O2, C20H24O2, C4H2FeO4

Molecular Weight

340.47 g/mol, 296.40 g/mol, 169.90 g/mol

Mechanism of Action

  • Inhibition of ovulation
  • Thickening of cervical mucus
  • Endometrial changes that discourage implantation

Indications

  • Contraception
  • Menstrual cycle regulation
  • Treatment of acne

Common Dosage Forms

  • Oral tablet

Typical Dosage

  • One tablet daily for 21 days, then no tablets for 7 days, followed by a new 28-day cycle.

Pediatric Dosage

  • Not recommended for children

Geriatric Dosage

  • May require a lower dosage in elderly patients

Side Effects

  • Nausea
  • Breast tenderness
  • Headaches
  • Irregular bleeding
  • Mood changes

Contraindications

  • Known or suspected pregnancy
  • History of blood clots
  • Breast cancer
  • Liver disease

Pregnancy Category

  • Category X - Contraindicated in pregnancy

Lactation Safety

  • Small amounts of hormonal components are excreted in breast milk, caution advised

Drug Interactions

  • Certain antibiotics
  • Anticonvulsants
  • St. John's Wort can reduce effectiveness

Overdose Symptoms

  • Nausea
  • Vomiting
  • Dizziness

Antidote for Overdose

  • No specific antidote, symptomatic treatment recommended

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Rapidly absorbed from the gastrointestinal tract
  • Distribution: Highly protein-bound
  • Metabolism: Hepatic metabolism
  • Excretion: Mainly excreted in urine and feces

Precautions

  • Smoking increases the risk of serious cardiovascular side effects
  • Regular monitoring of blood pressure advised

Warnings

  • Increased risk of cardiovascular events
  • Increased risk of blood clots

Others

  • Regular medical check-ups recommended for continued use