Lansoprazole

Generic Details

Generic Name

Lansoprazole

Other Names

  • Prevacid

Drug Class

  • Proton Pump Inhibitor

Chemical Formula

C16H14F3N3O2S

Molecular Weight

369.36 g/mol

Mechanism of Action

  • Inhibits the proton pump in the gastric parietal cell, suppressing the secretion of gastric acid.

Indications

  • Gastroesophageal Reflux Disease (GERD)
  • Peptic Ulcer Disease
  • Erosive Esophagitis
  • Zollinger-Ellison Syndrome

Common Dosage Forms

  • Capsules
  • Oral Suspension

Typical Dosage

  • 30 mg once daily for 4-8 weeks for most indications

Pediatric Dosage

  • Dosage based on weight and severity of condition - consult a pediatrician

Geriatric Dosage

  • Dosage adjustment may be needed based on renal function

Side Effects

  • Headache
  • Nausea
  • Diarrhea
  • Abdominal pain
  • Flatulence
  • Constipation

Contraindications

  • Hypersensitivity to lansoprazole
  • Severe liver disease

Pregnancy Category

  • Category B - no evidence of risk in humans

Lactation Safety

  • Safe to use while breastfeeding

Drug Interactions

  • Warfarin
  • Digoxin
  • Theophylline

Overdose Symptoms

  • Confusion
  • Blurred vision
  • Sweating
  • Increased heart rate

Antidote for Overdose

  • Symptomatic treatment and supportive measures

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Rapidly and completely absorbed after oral administration
  • Distribution: Widely distributed in the body
  • Metabolism: Primarily hepatic via CYP3A4
  • Excretion: Mainly via urine

Precautions

  • Monitor renal function in patients with impaired renal function

Warnings

  • May increase the risk of Clostridium difficile-associated diarrhea

Others