Levocarnitine

Generic Details

Generic Name

Levocarnitine

Other Names

  • L-Carnitine
  • L-Carnitine Tartrate

Drug Class

  • Amino Acid Derivative

Chemical Formula

C7H15NO3

Molecular Weight

161.20 g/mol

Mechanism of Action

  • Facilitates the transport of fatty acids into the mitochondria for energy production

Indications

  • Primary and secondary carnitine deficiencies
  • Chronic kidney disease requiring dialysis
  • Cardiac conditions
  • Cognitive impairments

Common Dosage Forms

  • Oral solution
  • Oral capsules
  • Injection

Typical Dosage

  • 500-2000 mg per day, depending on the condition being treated

Pediatric Dosage

  • Consult pediatrician for appropriate dosage

Geriatric Dosage

  • May require dosage adjustment based on renal function

Side Effects

  • Nausea
  • Vomiting
  • Diarrhea
  • Muscle cramps

Contraindications

  • Hypersensitivity to levocarnitine
  • Certain types of primary carnitine deficiency

Pregnancy Category

  • Category A - controlled studies in pregnant women have not shown a risk to the fetus

Lactation Safety

  • Compatible with breastfeeding

Drug Interactions

  • Thyroid hormones
  • Valproic acid
  • Warfarin

Overdose Symptoms

  • GI disturbances
  • Muscle weakness
  • Seizures

Antidote for Overdose

  • Discontinue medication and provide supportive care

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Well absorbed from the gastrointestinal tract
  • Distribution: Widely distributed in the body
  • Metabolism: Metabolized in the liver
  • Excretion: Excreted in urine

Precautions

  • Monitor renal function during long-term therapy
  • Adjust dosage in patients with renal impairment

Warnings

  • May interact with other medications, consult healthcare provider before starting levocarnitine

Others

  • May enhance exercise performance in some individuals