Ampicillin Sodium

Generic Details

Generic Name

Ampicillin-Sodium

Other Names

  • Ampicillin Sodium

Drug Class

  • Penicillin Antibiotic

Chemical Formula

C16H19N3O4S.Na

Molecular Weight

371.4 g/mol

Mechanism of Action

  • Inhibits bacterial cell wall synthesis by binding to penicillin-binding proteins (PBPs)

Indications

  • Bacterial infections such as respiratory tract infections, urinary tract infections, septicemia, meningitis, endocarditis, etc.

Common Dosage Forms

  • Capsules
  • Oral suspension
  • Injection

Typical Dosage

  • 250-500mg every 6 hours

Pediatric Dosage

  • Dose based on weight and severity of infection

Geriatric Dosage

  • May require lower doses due to reduced renal function

Side Effects

  • Diarrhea
  • Nausea
  • Rash
  • Allergic reactions
  • Superinfection

Contraindications

  • Hypersensitivity to penicillins
  • Infectious mononucleosis

Pregnancy Category

  • B - usually considered safe

Lactation Safety

  • Compatible with breastfeeding

Drug Interactions

  • Probenecid (decreases renal excretion)

Overdose Symptoms

  • Seizures
  • Confusion
  • Renal failure

Antidote for Overdose

  • Supportive care

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Well-absorbed orally
  • Distribution: Penetrates well into tissues and body fluids
  • Metabolism: Partially metabolized in the liver
  • Excretion: Primarily renal excretion

Precautions

  • Monitor for allergic reactions
  • Consider dose adjustments in renal impairment

Warnings

  • Risk of superinfection with prolonged use

Others

  • Complete the full course of antibiotics to prevent antibiotic resistance