Naproxen Sodium

Generic Details

Generic Name

Naproxen-Sodium

Other Names

  • Anaprox
  • Naprelan
  • Naprosyn
  • Aleve

Drug Class

  • Nonsteroidal Anti-Inflammatory Drug (NSAID)

Chemical Formula

C14H13NaO3

Molecular Weight

252.24 g/mol

Mechanism of Action

  • Inhibits the enzyme cyclooxygenase, leading to decreased prostaglandin synthesis

Indications

  • Pain relief
  • Fever reduction
  • Inflammatory conditions such as arthritis

Common Dosage Forms

  • Tablet
  • Suspension
  • Extended-release tablet
  • Liquid-filled capsule

Typical Dosage

  • 250-500 mg every 12 hours

Pediatric Dosage

  • Not recommended for children under 2 years old

Geriatric Dosage

  • Lower doses or longer dosing intervals may be required

Side Effects

  • Stomach upset
  • Ulcers
  • Kidney problems
  • High blood pressure

Contraindications

  • Hypersensitivity to naproxen or other NSAIDs
  • Active peptic ulcer disease

Pregnancy Category

  • Category C - Risk cannot be ruled out

Lactation Safety

  • Limited data available, caution advised

Drug Interactions

  • Aspirin
  • Anticoagulants
  • Lithium
  • Diuretics

Overdose Symptoms

  • Nausea
  • Vomiting
  • Headache
  • Dizziness
  • Gastric bleeding

Antidote for Overdose

  • Activated charcoal
  • Supportive care

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Rapid and complete
  • Distribution: Crosses the placenta, enters breast milk
  • Metabolism: Mainly hepatic
  • Excretion: Primarily renal

Precautions

  • Avoid in patients with a history of asthma
  • Use with caution in the elderly or patients with renal impairment

Warnings

  • Increased risk of cardiovascular events
  • May increase the risk of serious gastrointestinal adverse events

Others

  • Avoid alcohol consumption while taking naproxen