Omega-3 Acid Ethyl Esters

Generic Details

Generic Name

Omega-3-Acid-Ethyl-Esters

Other Names

  • Fish Oil
  • Epanova
  • Lovaza

Drug Class

  • Lipid-regulating agent

Chemical Formula

Molecular Weight

Mechanism of Action

  • Omega-3-Acid-Ethyl-Esters are polyunsaturated fatty acids that work by reducing the production of triglycerides in the liver.

Indications

  • Treatment of severe hypertriglyceridemia
  • Adjunct to diet in severe hypertriglyceridemia

Common Dosage Forms

  • Capsules

Typical Dosage

  • 4 grams per day, taken as a single dose or divided into two doses

Pediatric Dosage

  • Safety and efficacy not established in children

Geriatric Dosage

  • Dose adjustment may be necessary in older adults with impaired liver or kidney function

Side Effects

  • Common side effects include diarrhea, nausea, abdominal pain, and dyspepsia.
  • Rare but serious side effects may include pancreatitis and allergic reactions.

Contraindications

  • Hypersensitivity to fish or shellfish

Pregnancy Category

  • Category C - Safety in pregnancy has not been established, benefits should outweigh risks

Lactation Safety

  • Caution advised, unknown excretion into human milk

Drug Interactions

  • May increase the risk of bleeding when taken with anticoagulants

Overdose Symptoms

  • No specific overdose symptoms reported

Antidote for Overdose

  • No specific antidote, treatment is supportive

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Well absorbed from the gastrointestinal tract
  • Distribution: Distributed into plasma and erythrocyte lipids
  • Metabolism: Metabolized in the liver
  • Excretion: Mainly excreted in the feces

Precautions

  • Monitor liver function tests periodically during therapy

Warnings

  • Should not be used to treat high cholesterol levels if not associated with high triglyceride levels

Others