Pemirolast Potassium

Generic Details

Generic Name

Pemirolast-Potassium

Other Names

  • Pemirolast

Drug Class

  • Mast cell stabilizer
  • Antiallergic agent

Chemical Formula

C10H8KNO6S

Molecular Weight

305.35 g/mol

Mechanism of Action

  • Inhibits the release of histamine and other inflammatory mediators from mast cells

Indications

  • Allergic conjunctivitis
  • Prevention of asthma attacks triggered by allergens

Common Dosage Forms

  • Ophthalmic solution

Typical Dosage

  • 1-2 drops in the affected eye(s) 4 times daily

Pediatric Dosage

  • Safety and efficacy not established in children under 3 years old

Geriatric Dosage

  • No dosage adjustments necessary

Side Effects

  • Burning or stinging in the eyes
  • Headache
  • Blurry vision

Contraindications

  • Hypersensitivity to pemirolast-potassium or any component

Pregnancy Category

  • Category C - Risk cannot be ruled out

Lactation Safety

  • Use with caution, consult healthcare provider

Drug Interactions

  • No significant drug interactions reported

Overdose Symptoms

  • Not well-documented

Antidote for Overdose

  • No specific antidote, symptomatic treatment

Storage Conditions

  • Store at room temperature (15-30°C)

Pharmacokinetics

  • Absorption: Minimally absorbed after ophthalmic administration
  • Distribution: Limited systemic distribution
  • Metabolism: Metabolized in the liver
  • Excretion: Primarily through the urine

Precautions

  • Avoid contact lens wear during treatment
  • Do not use in the presence of eye infections

Warnings

  • Discontinue use if irritation or allergic reaction occurs

Others