Pivmecillinam

Generic Details

Generic Name

Pivmecillinam

Other Names

  • Pivampicillin

Drug Class

  • Antibiotic
  • Penicillin

Chemical Formula

C16H17N3O6S

Molecular Weight

371.39 g/mol

Mechanism of Action

  • Inhibits bacterial cell wall synthesis by binding to penicillin-binding proteins (PBPs)

Indications

  • Urinary tract infections
  • Respiratory tract infections
  • Skin and soft tissue infections

Common Dosage Forms

  • Tablet
  • Capsule

Typical Dosage

  • 200-400 mg every 6 hours

Pediatric Dosage

  • Dosing based on weight and age, to be determined by a healthcare provider

Geriatric Dosage

  • Lower doses may be required due to reduced renal function

Side Effects

  • Nausea
  • Vomiting
  • Diarrhea
  • Allergic reactions like rash or hives

Contraindications

  • Hypersensitivity to penicillins or beta-lactam antibiotics

Pregnancy Category

  • Safe for use in pregnancy

Lactation Safety

  • Considered safe during lactation

Drug Interactions

  • Probenecid may increase levels of pivmecillinam

Overdose Symptoms

  • Severe nausea
  • Vomiting
  • Diarrhea

Antidote for Overdose

  • Supportive care and monitoring

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Well-absorbed orally
  • Distribution: Distributed widely in body tissues
  • Metabolism: Partially metabolized in the liver
  • Excretion: Primarily excreted unchanged in the urine

Precautions

  • Use with caution in patients with renal impairment

Warnings

  • Risk of allergic reactions in patients with penicillin allergy

Others