Rabeprazole Sodium

Generic Details

Generic Name

Rabeprazole Sodium

Other Names

  • Rabeprazole

Drug Class

  • Proton Pump Inhibitor

Chemical Formula

C18H20N3NaO3S

Molecular Weight

381.42 g/mol

Mechanism of Action

  • Blocks the proton pump in gastric parietal cells, reducing gastric acid secretion

Indications

  • Gastroesophageal reflux disease (GERD)
  • Peptic ulcer disease
  • Zollinger-Ellison syndrome
  • Erosive esophagitis

Common Dosage Forms

  • Tablet
  • Delayed-release capsule

Typical Dosage

  • 20 mg once daily before a meal

Pediatric Dosage

  • Safety and efficacy not established in children

Geriatric Dosage

  • No dosage adjustment necessary in the elderly

Side Effects

  • Headache
  • Nausea
  • Abdominal pain
  • Diarrhea
  • Constipation

Contraindications

  • Hypersensitivity to rabeprazole
  • Co-administration with rilpivirine-containing products

Pregnancy Category

  • Category B

Lactation Safety

  • Probably safe to use during breastfeeding

Drug Interactions

  • Warfarin
  • Ketoconazole
  • Digoxin

Overdose Symptoms

  • Confusion
  • Drowsiness
  • Blurred vision

Antidote for Overdose

  • No specific antidote; provide supportive care

Storage Conditions

  • Store at room temperature away from moisture and heat

Pharmacokinetics

  • Absorption: Rapidly absorbed from the gastrointestinal tract
  • Distribution: Extensively bound to plasma proteins
  • Metabolism: Primarily metabolized in the liver
  • Excretion: Excreted in urine and feces

Precautions

  • Monitor magnesium levels in long-term use
  • Avoid abrupt discontinuation

Warnings

  • Increased risk of Clostridium difficile-associated diarrhea
  • Potential risk of osteoporosis-related fractures

Others